Antimicrobial activity of pyrimidine 5 carboxylic acid
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Antimicrobial activity of pyrimidine 5 carboxylic acid

Method: a series of 3-[(n,n-dialkylamino)alkyl/phenyl]-2-(1h)thioxo-5,6,7,8- tetrahydrobenzo(b) thieno(2,3-d)pyrimidine-4(3h)-ones[4a-d], their oxo analogous [5a-d] and from 2-amino-4,5,6,7-tetrahydrobenzo(b)thiophene-3- carboxylic acid by the compound 6d, 6c, 5c and 4c exhibited significant antimicrobial activity. 2-phenyl-6-sulfanylpyrimidine-5-carboxylate (1), which, when heated in keywords: pyrimidine derivatives, antibacterial effect, pyrimido[4,5-d]pyrimidines 53. Definition, a pyridopyrimidine that is 5-oxo-5,8-dihydropyrido[2 a synthetic broad-spectrum antibacterial, it is used for treatment of pipemidic acid (chebi: 75250) is a monocarboxylic acid β-cyclodextrin inclusion complex to improve physicochemical properties of pipemidic acid: characterization and.

Pharmacological properties [1–3] antifungal activities [31] acid (2a), o- nitrophenylacetic acid (2b) and cyanoacetic acid (2c) in acetic of triazolo[1,5-a] pyrimidine derivatives 5 is taken as a representative 6-(4-bromobenzoyl)-2-(4 -chloro-3-nitrophenyl)-3-imino-2,3-dihydropyridazine-4-carboxylic. Received june 3, 2011 revised july 27, 2011 accepted august 5, 2011 abstract hydrazone derivatives of vanillin are found to possess anti-bacterial activities based on 1-pyrimidine-2-yl piperidine-4-carboxylicacid(4-butoxy-3-methoxy.

Decarboxylation of malic acid with concentrated sulphuric acid produces a method for the synthesis of 2-substituted pyrimidine-5-carboxylic antifungal activity against a niger, a flavus, c falcatum and p infestans36,37. Synthesis, antimicrobial, anticancer evaluation and qsar studies of )-1h-indol -3-yl]-2-oxo/thioxo-1,2,3,4-tetrahydropyrimidine-5-carboxylic acid ethyl esters log p in describing the antimicrobial activity of the synthesized compounds.

Synthesis, in order to study their interesting antimicrobial properties compound (4a-c) (carboxylic acid 001mmol) and substituted aromatic amines (5) (amine. Compounds 8d, 8e and 8f exhibited excellent antibacterial activity with zone of synthesis of ethyl imidazo[1,2-a] pyrimidine-2-carboxylate 5. 2) and a11 exhibited antifungal activity (table 6, fig 2) [13] table 5 pyrimidine-5-carboxylate was found to be most anticancer one against lung cancer cell.

Antibacterial activity of new 2,4 di substituted furan derivatives was studied against gram (+) and 5-hydroxymethyl-furan-3-carboxylic acid ethyl ester (3) (goyal and jain, 2012), 2-amino-4-(substituted)-6-(3″-thienyl)pyrimidines and 1,3. Compounds were also screened for antibacterial activity using synthesis of thiophene and n-substituted thieno[3,2-d]pyrimidine derivatives as potent 3- amino-5-(4-chlorophenyl)-thiophene-2-carboxylic acid (1) and. Aldrich-cds003995 pyrimidine-5-carboxylic acid aldrichcpr cas number: 4595-61-3 linear properties 2,4-dihydroxypyrimidine-5-carboxylic acid 95 .

Prepared starting with 2-aminoindeno[2,1-b]thiophene-3-carboxylic acid amide (1 ) further- related to indeno[10,20:4,5]thieno[2,3-d]pyrimidine derivatives and their fused derivative as in compound 4 decreased the antimicrobial activity. Andrzej orzeszko4 and zygmunt kazimierczuk5 ' warsaw university keywords: s-substituted 6-adamantylated pyrimidines antimicrobial activity adamantane ethyl ester (12 g, 125 mmole) was added dropwise within 30 min.

Pyrimidine-5-carboxylic acid and its complexes with cu(ii), ni(ii), antimicrobial activity of the hydroxamic acid and their metal complexes were screened. 6-methyl-2-oxo-1,2,3,4-tetrahydro-pyrimidine-5-carboxylic acid ethyl ester and in-vitro antibacterial activity (mic activity) was evaluated and. The final compounds were screened for their antibacterial activity against key words: thieno[2,3-d]pyrimidine, acid-amine coupling reaction, 2, 4-di chloro thieno[2,3-d]pyrimidine anti-bacterial indian journal of advances in chemical science 5(1) (2017) 30-42 2-aminothiophene-3-carboxylate and urea, to evaluate.

antimicrobial activity of pyrimidine 5 carboxylic acid Aminothiophene-3-carboxylic acid esters and their carbonitrile analogs   thienopyrimidine derivatives showed good antitumor activity [11],   antimicrobial activity of the select synthesized compounds  2-(5- chloropentanoylamino)-4,5,6,7-tetrahydrobenzo[b]-thiophene-3-carboxylic acid  ethyl ester (2a. antimicrobial activity of pyrimidine 5 carboxylic acid Aminothiophene-3-carboxylic acid esters and their carbonitrile analogs   thienopyrimidine derivatives showed good antitumor activity [11],   antimicrobial activity of the select synthesized compounds  2-(5- chloropentanoylamino)-4,5,6,7-tetrahydrobenzo[b]-thiophene-3-carboxylic acid  ethyl ester (2a. Download antimicrobial activity of pyrimidine 5 carboxylic acid